JWH-251

Chemistry

Also known as

• 864445-39-6
• 55H9NDH32M
• 2-(2-Methylphenyl)-1-(1-pentyl-1H-indol-3-yl)ethanone
• DTXSID80235555
• RefChem:150690
• DTXCID10158046
• 1-Pentyl-3-(2-methylphenylacetyl)indole
• JWH 251

Attribution

• JW

  John W. Huffman — first synthesis, 2005

  1-Pentyl-3-(2-methylphenylacetyl)indole; Ki 29 nM CB1, 146 nM CB2, about 5x CB1-selective. Part of the 2005 phenylacetylindole series that mapped how ortho substituents on the phenylacetyl ring change receptor preference.

  source